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Hi-Tech Estrogenex
90 Tablets - Write a Review
By: Hi-Tech
Description
ESTROGENEX - A NATURAL AROMATASE INHIBITOR
AND ESTROGEN BLOCKER
ESTROGENEX - is a nutritional supplement,
available without a prescription, designed to
normalize all hormone levels, yielding a wide
spectrum of health and anti-aging benefits.
ESTROGENEX - is a multi-pathway
formulation that minimizes or eliminates the
undesirable effects associated with an estrogen
dominant environment.
ESTROGENEX - maintains the
correct testosterone to estrogen ratios that
yield the benefits associated with normal
estrogen levels.
ESTROGENEX - acts as an irreversible
anti-aromatase agent and is thus a powerful
elevator of total testosterone and maximum
liberator of free testosterone.
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ESTROGENEX - may also play
a role in long-term selective estrogen blocking
and/or inhibition of selective estrogen signaling.
ESTROGENEX - may contribute
to notable improvements in muscular growth and
fat loss, in addition to its wide array of health
and anti-aging benefits.
ESTROGENEX - is designed for:
Normalization of all hormone levels, with specific
tendencies toward testosterone dominance, in
all aging males.
Prevention and reversal of Gynecomastia.
Adjunctive supplementation for men undergoing
hormone replacement therapy to ensure that raising
testosterone levels will not yield an undesirable
increase in estrogen levels.
A natural, more effective alternative for traditional
testosterone hormone replacement therapy.
Bodybuilders and athletes during and immediately
after periods of anabolic steroid use for the
purpose of stimulating endogenous testosterone
production.
Testosterone: Free-Testosterone and Plasma Protein-Bound
Testosterone
Testosterone exists in the blood in either an
active (free) or unbound state (+-2%) or inactive
state bound to one of two proteins: sex-hormone-binding-globulin
(SHBG) (+-45%) or albumin (+-53%). Only when
testosterone is in its free state can it directly
interact with cellular receptors and exert its
activity. SHBG preferentially binds to testosterone
over estrogen. Higher levels of SHBG in women
help to maintain higher estrogen to testosterone
ratios. Increased estrogen leads to an increase
in SHBG. Thus, lowering the level of SHBG allows
for an increased level of free testosterone.
Obviously, if testosterone finds it more difficult
to locate available plasma proteins in the presence
of the additional compound, more will be left
in an unbound state.
The amount of free testosterone can be altered
(increased) by the use of aromatase inhibitors
(the less testosterone that is synthesized [aromatized]
into estrogen, the more total testosterone)
or inhibitors of the plasma proteins that bind
into testosterone. Manipulating the tendency
of a testosterone to exist in an unbound state
is an effective way to alter the overall activity
and potency of one?s overall testosterone levels.
Higher levels of testosterone produce an enhanced
anti-glucocorticoid effect, which yields an
anti-catabolic, or more precisely, anti-proteoolytic,
effect on muscle cells. This indirect anabolic
effect is the result of testosterone?s high
affinity for binding with glucocorticoid receptors,
thus blocking the normal messenger pathway that
triggers protein release from muscle tissue.
More free testosterone also likely results in
higher concentrations of IGF-1 and IGF-1 receptor
sites in skeletal muscle tissue. Correspondingly,
lower testosterone also likely yields less IGF-1
production and a corresponding decrease in IGF-1
receptor sites. Lower free testosterone also
likely means a weaker immune system.
The Synthesis (Aromatization) of Testosterone
to Estrogen in Males and the Significance of
Maintaining Correct Testosterone to Estrogen
Ratios.
Although testosterone is considered to be a
male hormone and estrogen a female hormone,
both hormones exist in both males and females
and serve important functions for both. Estrogen
is a term that really represents a collection
of female hormones, with esterone predominating.
Since esterone is the estrogen that is normally
in the highest concentration, it is an excellent
marker for basic estrogen levels for that reason.
At least three estrogens have multiple and overlapping
functions. Men obtain their estrogen through
the action of the aromatase, which synthesizes
(aromatizes) testosterone into estrogen. However,
when concentrations of estrogen become too high
and/or the normal ratio of testosterone to estrogen
decreases, the potential for the development
of undesirable conditions arises. This includes
the development of the female breast tissue
(gynecomastia), increased body fat and water
retention. Also, research suggests that DHT
and prostate tissue growth have a direct connection
to above normal estrogen elevations and reduced
testosterone levels.
The ESTROGENEX
- Mechanism of Action
The ESTROGENEX - proprietary formula was developed
by combining naturally occurring aromatase inhibitors
and inhibitors of the action of SHBG. The primary
active ingredients in ESTROGENEX are Coumesterol
and Chrysin. ESTROGENEX does not exert its action
through any direct hormonal or prohormonal activity
(androgenic or estrogenic).
Before ESTROGENEX , little
success had been achieved using chrysin as an
effective aromatase inhibitor because chrysin
is poorly absorbed in the bloodstream. However,
in addition to their own specific aromatase
inhibiting and estrogen blocking actions, the
proprietary blend of other ingredients work
in synergy with chrysin to maintain a stable
estrogen environment. We also incorporated our
proprietary delivery system called EXTEND-RX?
to avoid competing with other hormones such
as testosterone in the Aromatase Cytochrome
P450.
It is believed that ESTROGENEX exerts its effects
through several mechanisms of action, which
can be classified into two groups: 1. as an
inhibitor of the aromatase enzyme responsible
for the conversion of testosterone to estrogen
and an inhibitor of the action of SHBG, and
2. as a blocker of selective anabolic estrogen
receptors and/or inhibitor of selective estrogen
signaling.
Substances that are aromatase inhibitors block
the action of the enzyme aromatase that converts
testosterone to estrogen. Substances that act
as an anti-estrogen are those that block the
estrogen receptor. Thus, even though there is
estrogen circulating in the blood, the estrogen
cannot exert its effects because it is blocked
from attaching to its estrogen receptor. The
dietary supplement ESTROGENEX ? is a multi-pathway
agent that exerts its influence by blocking
various stages in the aromatase process and
by inhibiting SHBG's action; an activity not
clearly addressed by any of the aromatase inhibiting
or anti-estrogen products. Further, it appears
that use of ESTROGENEX may result in long-term
blocking of selective anabolic estrogen receptors
and/or inhibition of selective estrogen signaling
(these anabolic estrogens are those demonstrating
the undesirable effects associated with breast
cancer and gynecomastia). This activity has
not been addressed by any known dietary supplements
or pharmacological agents.
ESTROGENEX
as an Elevator of Total Testosterone and Liberator
of Free Testosterone
As a powerful aromatase inhibitor, ESTROGENEX
also possesses notable testosterone stimulating
properties. The aromatase inhibiting action
reduces the signal that estrogen sends to the
brain to suppress endogenous testosterone production
(estrogen is a main feedback signal to control
the release of testosterone, thus increasing
the testicular output of testosterone). ESTROGENEX
thus assists in resetting the body's level of
its own natural testosterone production by regulating
the activity of the hypothalamic-pituitary-testicular
axis (HPTA), which constantly adjusts the body's
production of testosterone to maintain target
blood levels. Continued use of ESTROGENEX results
in not only a significant reduction in the production
of estrogen, but also a corresponding substantial
increase in endogenous testosterone.
Only ESTROGENEX addresses all
possible channels to estrogen maintenance and
free testosterone elevation, which means optimal
hormonal levels for muscle building, fat loss
and anti-aging support.
Supplement Facts
One tablets supply the following ingredients:
Servings Per Container: 90
Proprietary Blend - 600mg
with Extend-RX Technology
(Chrysin 99%, Green Tea RM7343 Extract (leaves),
Beta-Sitosterol 90%, Muira Puama Extract (root),
Quercitin, Soy ISO Flavone 40% (flavanoid),
Coumesterol (flavanoid), 6, 7 Dihydroxybergamottin
(fruit), Naringen (fruit).)
Other Ingredients:
Microcrystalline Cellulose, Starch, Stearic
Acid, Sodium Starch Glycolate, Triacetin, Silica,
FD & C Red #3, FD & C Yellow #6
Directions
Take three tablets of Estrogenex daily. Estrogenex
is best taken near mealtime.
* No claims found on this web page or in print have been evaluated by the Food and Drug Administration. This product is not intended to diagnose, treat, cure, or prevent any disease. No claim or opinion about weight loss, bodybuilding or general health on this web page is intended to be, nor should be construed to be, medical advice. Please consult with a healthcare professional before starting any weight loss diet or exercise program.
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